| Gene | No. Representative PDBs | No. Target Structures | No. Pockets |
|---|---|---|---|
| ABL1 | 6 | 6 | 27 |
| ACAA1 | 1 | 1 | 3 |
| ACACA | 2 | 2 | 8 |
| ACACB | 2 | 2 | 8 |
| ACAD8 | 1 | 1 | 3 |
| ACADS | 1 | 1 | 4 |
| ACADSB | 1 | 1 | 3 |
| ACAT1 | 1 | 1 | 3 |
| ACTN1 | 1 | 1 | 3 |
| ACVR1 | 3 | 3 | 15 |
| ACY1 | 1 | 2 | 5 |
| ADA | 1 | 1 | 5 |
| ADAM17 | 1 | 1 | 5 |
| ADAR | 2 | 2 | 9 |
| ADCK3 | 1 | 1 | 5 |
| ADI1 | 1 | 1 | 5 |
| ADRB2 | 2 | 2 | 9 |
| ADSL | 1 | 1 | 5 |
| AFF4 | 1 | 1 | 2 |
| AGT | 1 | 1 | 5 |
| AGTR1 | 1 | 1 | 1 |
| AHCY | 1 | 1 | 5 |
| AIFM1 | 1 | 1 | 1 |
| AIM2 | 3 | 3 | 11 |
| AIMP2 | 2 | 2 | 5 |
| AK1 | 1 | 1 | 3 |
| AK3 | 1 | 1 | 3 |
| AK4 | 3 | 3 | 5 |
| AKR1A1 | 1 | 1 | 5 |
| AKR1B1 | 1 | 1 | 4 |
| AKR1C2 | 1 | 1 | 3 |
| AKR7A2 | 1 | 1 | 3 |
| AKT1 | 3 | 3 | 12 |
| AKT2 | 1 | 1 | 5 |
| AKT3 | 1 | 1 | 2 |
| ALB | 2 | 2 | 10 |
| ALDH18A1 | 1 | 1 | 4 |
| ALDH1A1 | 1 | 1 | 2 |
| ALDH2 | 1 | 1 | 4 |
| ALDH4A1 | 2 | 2 | 8 |
| ALDH5A1 | 1 | 1 | 3 |
| ALDH7A1 | 1 | 1 | 1 |
| ALDOC | 1 | 1 | 3 |
| ALK | 2 | 2 | 5 |
| AMBP | 2 | 2 | 5 |
| AMD1 | 1 | 1 | 5 |
| AMT | 1 | 1 | 3 |
| ANXA2 | 2 | 2 | 8 |
| ANXA3 | 1 | 1 | 5 |
| ANXA5 | 1 | 1 | 5 |
| AOC3 | 1 | 1 | 5 |
| AP1B1 | 2 | 2 | 8 |
| APC | 5 | 5 | 17 |
| APEX1 | 1 | 1 | 5 |
| APOA1 | 3 | 3 | 10 |
| APOE | 1 | 1 | 5 |
| APOH | 3 | 3 | 14 |
| APOM | 1 | 1 | 5 |
| APP | 7 | 7 | 26 |
| APRT | 1 | 1 | 3 |
| AR | 1 | 1 | 3 |
| ARF1 | 3 | 3 | 13 |
| ARF4 | 1 | 1 | 5 |
| ARFIP2 | 2 | 2 | 8 |
| ARG1 | 1 | 1 | 5 |
| ARG2 | 1 | 1 | 5 |
| ARHGAP1 | 2 | 2 | 10 |
| ARHGAP9 | 1 | 1 | 5 |
| ARHGDIB | 1 | 1 | 4 |
| ARHGEF12 | 2 | 2 | 10 |
| ARL1 | 1 | 1 | 5 |
| ARNT | 1 | 1 | 5 |
| ASF1A | 1 | 1 | 5 |
| ASH2L | 4 | 4 | 13 |
| ASL | 1 | 1 | 4 |
| ASMTL | 1 | 1 | 5 |
| ASPH | 1 | 1 | 4 |
| ASS1 | 1 | 1 | 3 |
| ATF2 | 1 | 1 | 4 |
| ATG12 | 1 | 1 | 5 |
| ATG4A | 1 | 1 | 5 |
| ATG4B | 1 | 1 | 5 |
| ATG5 | 2 | 2 | 10 |
| ATOX1 | 1 | 1 | 2 |
| ATP7A | 1 | 1 | 5 |
| AXL | 1 | 1 | 4 |
| B2M | 10 | 10 | 40 |
| B3GAT3 | 1 | 1 | 2 |
| BACE1 | 3 | 3 | 4 |
| BACE2 | 1 | 1 | 1 |
| BACH1 | 1 | 1 | 5 |
| BACH2 | 1 | 1 | 4 |
| BAG1 | 2 | 2 | 10 |
| BAG6 | 2 | 2 | 7 |
| BAK1 | 3 | 3 | 11 |
| BAZ2B | 3 | 3 | 11 |
| BBC3 | 1 | 1 | 2 |
| BBS9 | 1 | 1 | 1 |
| BCAR1 | 2 | 2 | 10 |
| BCAT1 | 1 | 1 | 3 |